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Found 1 Enz. Inhib. hit(s) with Target = 'Histone deacetylase 1' and Ligand = 'BDBM27775'
TargetHistone deacetylase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM27775(N-[2-amino-5-(thiophen-3-yl)phenyl]-4-{1,8-diazasp...)
Affinity DataIC50:  8nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed