TargetHistone deacetylase 5(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus
Curated by ChEMBL
Birla Institute Of Technology And Science-Pilani Hyderabad Campus
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human HDAC5 using fluorescent as substrate measured for 30 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus
Curated by ChEMBL
Birla Institute Of Technology And Science-Pilani Hyderabad Campus
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMpH: 8.0Assay Description:Activity against HDACs 1 to 11 was assessed by using an acetylated 7-amino-4-methylcoumarin (AMC)-labeled peptide substrate. A substrate based on res...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus
Curated by ChEMBL
Birla Institute Of Technology And Science-Pilani Hyderabad Campus
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human HDAC5 using Boc-Lys(trifluoroacetyl)-AMC) as substrate by fluorimetric assayMore data for this Ligand-Target Pair