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Found 3 Enz. Inhib. hit(s) with Target = 'Histone deacetylase 5' and Ligand = 'BDBM163619'
TargetHistone deacetylase 5(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM163619(UF010 | US10807944, Compound UF010 | US11731934, C...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human HDAC5 using fluorescent as substrate measured for 30 mins by fluorescence based microtiter plate assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM163619(UF010 | US10807944, Compound UF010 | US11731934, C...)
Affinity DataIC50: >1.00E+5nMpH: 8.0Assay Description:Activity against HDACs 1 to 11 was assessed by using an acetylated 7-amino-4-methylcoumarin (AMC)-labeled peptide substrate. A substrate based on res...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Birla Institute Of Technology And Science-Pilani Hyderabad Campus

Curated by ChEMBL
LigandPNGBDBM163619(UF010 | US10807944, Compound UF010 | US11731934, C...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human HDAC5 using Boc-Lys(trifluoroacetyl)-AMC) as substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed