Affinity DataKi: 25nMAssay Description:Competitive inhibition of HDAC5 using KI-104 as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 175nMAssay Description:Inhibition of human HDAC5More data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Tested in vitro for antagonist activity against H3 receptor of guinea pig jejunum.More data for this Ligand-Target Pair