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Found 4 Enz. Inhib. hit(s) with Target = 'Histone deacetylase 9' and Ligand = 'BDBM272140'
TargetHistone deacetylase 9(Homo sapiens (Human))
Chdi Foundation

US Patent
LigandPNGBDBM272140(E1-(abs)-2-(1,5-Dimethyl-1H-pyrazol-4-yl)-5-(3- fl...)
Affinity DataIC50:  68nMAssay Description:The potency of the compounds is quantified by measuring the Histone Deacetylase 9 (HDAC9) enzymatic activity using the fluorogenic substrate, Boc-Lys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 9(Homo sapiens (Human))
Chdi Foundation

US Patent
LigandPNGBDBM272140(E1-(abs)-2-(1,5-Dimethyl-1H-pyrazol-4-yl)-5-(3- fl...)
Affinity DataIC50:  68nMAssay Description:The potency of the compounds is quantified by measuring the Histone Deacetylase 9 (HDAC9) enzymatic activity using the fluorogenic substrate, Boc-Lys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 9(Homo sapiens (Human))
Chdi Foundation

US Patent
LigandPNGBDBM272140(E1-(abs)-2-(1,5-Dimethyl-1H-pyrazol-4-yl)-5-(3- fl...)
Affinity DataIC50:  200nMAssay Description:The potency of the compounds is quantified by measuring the Histone Deacetylase 9 (HDAC9) enzymatic activity using the fluorogenic substrate, Boc-Lys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 9(Homo sapiens (Human))
Chdi Foundation

US Patent
LigandPNGBDBM272140(E1-(abs)-2-(1,5-Dimethyl-1H-pyrazol-4-yl)-5-(3- fl...)
Affinity DataIC50:  200nMAssay Description:The potency of the compounds is quantified by measuring the Histone Deacetylase 9 (HDAC9) enzymatic activity using the fluorogenic substrate, Boc-Lys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent