Found 3 Enz. Inhib. hit(s) with Target = 'Homeodomain-interacting protein kinase 3' and Ligand = 'BDBM2579'
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 202nMAssay Description:Inhibition of human HIPK3 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 710nMAssay Description:Inhibition of human HIPK3 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 75nMAssay Description:Binding constant for HIPK3 kinase domainMore data for this Ligand-Target Pair