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Found 4 Enz. Inhib. hit(s) with Target = 'Hydroxycarboxylic acid receptor 2' and Ligand = 'BDBM50325899'
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325899(2-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4(3H)-on...)
Affinity DataIC50:  400nMAssay Description:Displacement of radioligand from rat GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325899(2-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4(3H)-on...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of radioligand from human GPR109AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325899(2-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4(3H)-on...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GPR109A receptor assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50325899(2-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4(3H)-on...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at rat GPR109A receptor assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed