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Compile Data Set for Download or QSAR
maximum 50k data
Found
1
Enz. Inhib. hit(s) with Target = 'Insulin receptor' and Ligand = 'BDBM2580'
Target
Insulin receptor
(Homo sapiens (Human))
Merck Research Laboratories
Ligand
BDBM2580
(K252a | methyl (15R,16S,18S)-16-hydroxy-15-methyl-...)
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Affinity Data
IC50: 210nM
pH: 7.4 T: 2°C
Assay Description:
The assay uses purified enzyme interacting with biotinylated peptide substrate.HTRF is based on the proximity of europium cryptate (donor fluorophore...
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