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Found 2 Enz. Inhib. hit(s) with Target = 'Insulin receptor [964-1370]' and Ligand = 'BDBM184542'
TargetInsulin receptor [964-1370](Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184542(US9150578, I-169 | US9150578, I-173)
Affinity DataIC50:  0.100nMpH: 7.4Assay Description:The kinase activity is measured by DELFIA.RTM. assay (dissociation-enhanced lanthanide fluorescence immunoassay, Perkin Elmer). The cytoplasmic kinas...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetInsulin receptor [964-1370](Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184542(US9150578, I-169 | US9150578, I-173)
Affinity DataIC50:  0.200nMpH: 7.4Assay Description:The kinase activity is measured by DELFIA.RTM. assay (dissociation-enhanced lanthanide fluorescence immunoassay, Perkin Elmer). The cytoplasmic kinas...More data for this Ligand-Target Pair
In DepthDetails US Patent