Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Integrase' and Ligand = 'BDBM50162325'
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162325(5-ethyl-3-{2-[1-(5-ethyl-2-sulfanyl-3-thienyl)-(E)...)
Affinity DataIC50:  6.00E+3nMAssay Description:Concentration to inhibit strand transfer of soluble mutant (F185K, C280S) of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162325(5-ethyl-3-{2-[1-(5-ethyl-2-sulfanyl-3-thienyl)-(E)...)
Affinity DataIC50:  2.10E+4nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162325(5-ethyl-3-{2-[1-(5-ethyl-2-sulfanyl-3-thienyl)-(E)...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162325(5-ethyl-3-{2-[1-(5-ethyl-2-sulfanyl-3-thienyl)-(E)...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of soluble mutant (F185K, C280S) of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed