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Found 2 Enz. Inhib. hit(s) with Target = 'Integrase' and Ligand = 'BDBM50162335'
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162335(5-Cyclopropyl-2H-pyrazole-3-carboxylic acid [1-(2,...)
Affinity DataIC50:  4.30E+4nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162335(5-Cyclopropyl-2H-pyrazole-3-carboxylic acid [1-(2,...)
Affinity DataIC50:  1.77E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed