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Found 2 Enz. Inhib. hit(s) with Target = 'Integrin alpha-4/beta-1' and Ligand = 'BDBM50111227'
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50111227((S)-3-(2',6'-Dimethoxy-biphenyl-4-yl)-2-(3,4-dioxo...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of binding of Very late antigen 4/vascular cell adhesion molecule 1 in a protein-based ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50111227((S)-3-(2',6'-Dimethoxy-biphenyl-4-yl)-2-(3,4-dioxo...)
Affinity DataIC50:  710nMAssay Description:Inhibition of binding of Very late antigen 4/vascular cell adhesion molecule 1 in a cell based ligand binding assay (Jurkat cells)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed