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Found 4 Enz. Inhib. hit(s) with Target = 'Interleukin-2 receptor subunit alpha' and Ligand = 'BDBM50147974'
TargetInterleukin-2 receptor subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50147974((S)-2-[2-((R)-1-Carbamimidoyl-piperidin-3-yl)-acet...)
Affinity DataIC50:  3.00E+3nMAssay Description:Antagonist activity at adrenergic Alpha-1D receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetInterleukin-2 receptor subunit alpha(Mus musculus)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50147974((S)-2-[2-((R)-1-Carbamimidoyl-piperidin-3-yl)-acet...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of mouse Interleukin-2 receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterleukin-2 receptor subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50147974((S)-2-[2-((R)-1-Carbamimidoyl-piperidin-3-yl)-acet...)
Affinity DataIC50:  6.00E+3nMAssay Description:Competitive inhibition of IL2 receptor alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-2 receptor subunit alpha(Mus musculus)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50147974((S)-2-[2-((R)-1-Carbamimidoyl-piperidin-3-yl)-acet...)
Affinity DataEC50:  1.00E+5nMAssay Description:Effective concentration required against phosphorylation of Mammary gland factor/STAT5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed