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Found 1 Enz. Inhib. hit(s) with Target = 'Kallikrein-14' and Ligand = 'BDBM50289001'
TargetKallikrein-14(Homo sapiens (Human))
Sixera Pharma

US Patent
LigandPNGBDBM50289001(2-(2-Iodo-phenyl)-6,7-dimethoxy-benzo[d][1,3]oxazi...)
Affinity DataKi:  2.10E+3nM ΔG°:  -33.7kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK14, Substrate S-2302 (Chromogenics, cat. no. 820340). KLK14 activity was determined at 37° C. in 0.1 mM Tris, pH ...More data for this Ligand-Target Pair
In DepthDetails US Patent