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Found 3 Enz. Inhib. hit(s) with Target = 'Kallikrein-5 [D153N]' and Ligand = 'BDBM50355086'
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50355086(CHEMBL1834753)
Affinity DataKi:  2.29E+4nMAssay Description:Competitive inhibition of human kallikrein-5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50355086(CHEMBL1834753)
Affinity DataKi:  2.44E+4nMAssay Description:Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50355086(CHEMBL1834753)
Affinity DataIC50:  7.29E+4nMAssay Description:Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by spectrofluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed