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Found 1 Enz. Inhib. hit(s) with Target = 'Kallikrein-7' and Ligand = 'BDBM113300'
TargetKallikrein-7(Homo sapiens (Human))
Sixera Pharma

US Patent
LigandPNGBDBM113300(US9695194, 16)
Affinity DataKi:  149nM ΔG°:  -40.5kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent