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Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM425899'
TargetKappa-type opioid receptor(Homo sapiens (Human))
Inheris Pharmaceuticals

US Patent
LigandPNGBDBM425899(US10512644, Compound alpha-6-mPEG5-O-Morphine)
Affinity DataKi:  558nMAssay Description:Briefly, serial dilutions of the test compounds were placed in a 96-well plate to which were added SPA beads, membrane and radioligand. The assay con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKappa-type opioid receptor(Homo sapiens (Human))
Inheris Pharmaceuticals

US Patent
LigandPNGBDBM425899(US10512644, Compound alpha-6-mPEG5-O-Morphine)
Affinity DataEC50:  2.30E+3nMAssay Description:Briefly, suspensions of cells expressing either the mu, kappa or delta opioid receptors were prepared in buffer containing 0.5 mM isobutyl-methyl xan...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent