Affinity DataKi: 61nMAssay Description:Binding affinity by its ability to displace [3H]-U-69,593 from kappa receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:In vivo binding affinity was evaluated by measuring the ability to displace [3H]U-69593 radioligand binding from Opioid receptor kappa 1 in guinea pi...More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity against Opioid receptor kappa 1 from guinea pig brain membranes using [3H]U-69593Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.09E+5nMAssay Description:Binding affinity determined by displacing [3H]U69,593 from Opioid receptor kappa 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 117nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human Opioid receptor kappa 1 ex...More data for this Ligand-Target Pair