Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50169777'
TargetKappa-type opioid receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169777((3S,4aR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,...)
Affinity DataKi:  1.30nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169777((3S,4aR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,...)
Affinity DataKi:  1.30nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169777((3S,4aR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,...)
Affinity DataEC50:  4.5nMAssay Description:Activation of human k-opioid receptor as increased [35S]GTPcS binding More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169777((3S,4aR,6S,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl-4a,...)
Affinity DataEC50:  4.5nMAssay Description:Activation of human k-opioid receptor as increased [35S]GTPcS binding More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed