Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50185316'
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50185316(CHEMBL3824309)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]diprenorphine from human KOR expressed in CHO cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50185316(CHEMBL3824309)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human KOR expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed