Affinity DataKi: 55nMAssay Description:Displacement of [3H]diprenorphine from k-Y312A-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 292nMAssay Description:Displacement of [3H]diprenorphine from k-E297A-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 488nMAssay Description:Displacement of [3H]diprenorphine from opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 588nMAssay Description:selective binding affinity against kappa opioid receptor, using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 588nMAssay Description:Displacement of [3H]U69493 from Hartley guinea pig kappa opioid receptor by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of [3H]-U-69,593 binding to Opioid receptor kappa 1 from mouse brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: >3.00E+3nMAssay Description:The compound tested for agonistic activity against Opioid receptor kappa 1 as the [3H]- U-69,594 radioligand.More data for this Ligand-Target Pair