Affinity DataKi: 0.490nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cell membranes incubated for 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]-HS665 from KOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 463nMAssay Description:Inhibition of kappa opioid receptor (unknown origin) assessed as increase in beta-arrestin 2 recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: 3.60nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cell membranes incubated for 60 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Inhibition of kappa opioid receptor (unknown origin) by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair