TargetKappa-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human KOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Julius Maximilian University Of W£Rzburg
Curated by ChEMBL
Affinity DataKd: 9.5nMAssay Description:Binding affinity to recombinant human KOR transiently expressed in CHOK1 cells measured after 20 mins by TIRF microscopic analysisMore data for this Ligand-Target Pair