Affinity DataKi: 0.0740nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.870nMAssay Description:Agonist activity at human KISS1R transfected in CHO cells assessed as intracellular calcium flux after 24 hrs by functional FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonist activity at rat KISS1R transfected in CHO cells assessed as intracellular calcium flux after 24 hrs by functional FLIPR assayMore data for this Ligand-Target Pair