Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'KiSS-1 receptor' and Ligand = 'BDBM50216076'
TargetKiSS-1 receptor(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50216076((2S)-2-{2-[(2S)-2-[(4-{[bis(pyridin-2-ylmethyl)ami...)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at GPR54 expressed in CHO cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed