Affinity DataKi: 0.0780nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0920nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0720nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair