Found 1 Enz. Inhib. hit(s) with Target = 'Kinesin-1 heavy chain/Proto-oncogene tyrosine-protein kinase receptor Ret' and Ligand = 'BDBM50601766'
TargetKinesin-1 heavy chain/Proto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
University Of Arkansas For Medical Sciences
Curated by ChEMBL
University Of Arkansas For Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of KIF5B-RET (unknown origin) assessed as inhibition of RET autophosphorylation expressed in mouse BaF3 cellsMore data for this Ligand-Target Pair