Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Kinesin-like protein KIF20B' and Ligand = 'BDBM50056904'
TargetKinesin-like protein KIF20B(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50056904(cid_65751 | 3,8-Dihydroxy-11-oxo-1-(2-oxo-heptyl)-...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of microtubule-stimulated ATPase activity of N-terminal His6-tagged/SUMO-fused human MPP1 motor domain (2 to 477 residues) expressed in Es...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2018
Entry Details Article
PubMed
TargetKinesin-like protein KIF20B(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50056904(cid_65751 | 3,8-Dihydroxy-11-oxo-1-(2-oxo-heptyl)-...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of microtubule-stimulated ATPase activity of N-terminal His6-tagged/SUMO-fused human MPP1 motor domain (57 to 491 residues) expressed in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2018
Entry Details Article
PubMed
TargetKinesin-like protein KIF20B(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50056904(cid_65751 | 3,8-Dihydroxy-11-oxo-1-(2-oxo-heptyl)-...)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of basal ATPase activity of N-terminal His6-tagged/SUMO-fused human MPP1 motor domain (57 to 491 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2018
Entry Details Article
PubMed
TargetKinesin-like protein KIF20B(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50056904(cid_65751 | 3,8-Dihydroxy-11-oxo-1-(2-oxo-heptyl)-...)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of basal ATPase activity of N-terminal His6-tagged/SUMO-fused human MPP1 motor domain (2 to 477 residues) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2018
Entry Details Article
PubMed