Found 5 Enz. Inhib. hit(s) with Target = 'L-lactate dehydrogenase A chain' and Ligand = 'BDBM50052248'
Affinity DataIC50: 880nMAssay Description:Inhibition of human recombinant carboxy-terminal His-tagged LDHA by MS endpoint assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:LDHA, LDHB, LDHC, MDH1 and MDH2 enzymatic assays have been described in detail previously [Dragovich, P.S. et al, Bioorg. Med. Chem. Lett. 24:3764-37...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human recombinant carboxy-terminal His-tagged LDHA by UV endpoint assayMore data for this Ligand-Target Pair
Affinity DataKd: 7.71E+5nMAssay Description:Inhibition of human recombinant carboxy-terminal His-tagged LDHA by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 3.50E+3nMAssay Description:Inhibition of human recombinant carboxy-terminal His-tagged LDHA by SPR assay in presence of +NADHMore data for this Ligand-Target Pair