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Found 3 Enz. Inhib. hit(s) with Target = 'Leucyl-cystinyl aminopeptidase' and Ligand = 'BDBM50331048'
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50331048(CHEMBL1277437 | ethyl 2-acetamido-7-hydroxy-4-(qui...)
Affinity DataKi:  20nMAssay Description:Inhibition of catalytic activity of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50331048(CHEMBL1277437 | ethyl 2-acetamido-7-hydroxy-4-(qui...)
Affinity DataKi:  20nMAssay Description:Inhibition of catalytic activity of recombinant human IRAP transfected in human HEK-293 cells assessed as clevage of substrate L-leucine-p-nitroanili...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50331048(CHEMBL1277437 | ethyl 2-acetamido-7-hydroxy-4-(qui...)
Affinity DataKi:  30nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed