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Found 2 Enz. Inhib. hit(s) with Target = 'Lysophosphatidic acid receptor 3' and Ligand = 'BDBM50398092'
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50398092(CHEMBL2182047 | US9321738, 5)
Affinity DataIC50:  6.30E+3nMAssay Description:Antagonist activity at human recombinant LPA3 expressed in chem-1 cells assessed as inhibition of LPA-induced intracellular calcium mobilization incu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50398092(CHEMBL2182047 | US9321738, 5)
Affinity DataIC50:  6.31E+3nMT: 2°CAssay Description:Test compounds were prepared by adding 90 μL of HBSS/20 mM HEPES/0.1% BSA buffer to 2 μL of serially diluted compounds. To prepare serial dilut...More data for this Ligand-Target Pair
In DepthDetails US Patent