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Found 2 Enz. Inhib. hit(s) with Target = 'MAP kinase-interacting serine/threonine-protein kinase 1' and Ligand = 'BDBM50079471'
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Ocean University Of China And Laboratory For Marine Drugs And Bioproducts

Curated by ChEMBL
LigandPNGBDBM50079471(CHEMBL3417198)
Affinity DataKi:  300nMAssay Description:Binding affinity to MNK1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Ocean University Of China And Laboratory For Marine Drugs And Bioproducts

Curated by ChEMBL
LigandPNGBDBM50079471(CHEMBL3417198)
Affinity DataKi:  4.82E+3nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed