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Found
1
Enz. Inhib. hit(s) with Target = 'MLL1-WRAD2 complex' and Ligand = 'BDBM552955'
Target
MLL1-WRAD2 complex
(Homo sapiens (Human))
Propellon Therapeutics
US Patent
Ligand
BDBM552955
(N-[5-[2-(cyclopropylamino) pyrimidin-5-yl]-4-fluor...)
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Affinity Data
IC50: 8.36E+3nM
Assay Description:
Compound potency was assessed through incorporation of 3H-SAM into oligonucleosomes purified from HeLa cells. Specifically, recombinant human MLL1 (a...
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Target Info
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Ligand Info
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