Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Mas-related G-protein coupled receptor member X2' and Ligand = 'BDBM224021'
TargetMas-related G-protein coupled receptor member X2(Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM224021(BAM8-22 | VGRPEWWMDYQKRYG)
Affinity DataEC50:  1.10E+4nMpH: 7.4 T: 2°CAssay Description:HTLA cells (HEK-T cells stably expressing a β-arrestin2-TEV fusion protein and a tTa-dependent luciferase reporter) were maintained in DMEM (Cor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X2(Homo sapiens (Human))
University Of North Carolina

LigandPNGBDBM224021(BAM8-22 | VGRPEWWMDYQKRYG)
Affinity DataEC50:  8.90E+3nMpH: 7.4 T: 2°CAssay Description:MRGPRX2 stable cells were maintained in DMEM containing 10% FBS, 100 μg/ml hygromycin B, and 15 μg/ml blasticidin. For the calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed