Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50193603'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193603((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-(triflu...)
Affinity DataIC50:  1.30nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193603((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-(triflu...)
Affinity DataIC50:  1.30nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193603((E)-N-(4-amino-2-propylquinolin-6-yl)-3-(4-(triflu...)
Affinity DataEC50:  61nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed