Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50193621'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193621((E)-N-(2-propyl-4-(pyrrolidin-1-yl)quinolin-6-yl)-...)
Affinity DataIC50:  17nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193621((E)-N-(2-propyl-4-(pyrrolidin-1-yl)quinolin-6-yl)-...)
Affinity DataEC50:  2.80E+3nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed