Affinity DataKi: 690nMAssay Description:Binding affinity against human Melanocortin 3 receptor by gamma-MCH displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 3 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
Affinity DataEC50: 520nMAssay Description:Effective concentration for intracellular cAMP accumulation in human melanocortin 3 receptor expressing HEK 293 cells; (N = 4)More data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Intracellular cAMP accumulation in human Melanocortin 3 receptor functional assay.More data for this Ligand-Target Pair