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Found 4 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 3' and Ligand = 'BDBM50314764'
TargetMelanocortin receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314764(CHEMBL1093304 | trans-N-(2-((R)-1'-((3S,4R)-1-tert...)
Affinity DataIC50:  890nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC3R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314764(CHEMBL1093304 | trans-N-(2-((R)-1'-((3S,4R)-1-tert...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at mouse MC3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314764(CHEMBL1093304 | trans-N-(2-((R)-1'-((3S,4R)-1-tert...)
Affinity DataEC50:  997nMAssay Description:Agonist activity at rat MC3R expressed in CHO cells assessed as stimulation of intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50314764(CHEMBL1093304 | trans-N-(2-((R)-1'-((3S,4R)-1-tert...)
Affinity DataEC50:  351nMAssay Description:Agonist activity at human MC3R expressed in CHO cells assessed as stimulation of intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed