Affinity DataIC50: 52nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 82nMAssay Description:Effective concentration towards human melanocortin-4 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair