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Found 3 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50157314'
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157314((S)-4-Methyl-piperazine-2-carboxylic acid [(R)-2-(...)
Affinity DataIC50:  7nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157314((S)-4-Methyl-piperazine-2-carboxylic acid [(R)-2-(...)
Affinity DataIC50:  7nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157314((S)-4-Methyl-piperazine-2-carboxylic acid [(R)-2-(...)
Affinity DataEC50:  11nMAssay Description:Effective concentration towards human melanocortin-4 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed