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Found 2 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50250586'
TargetMelanocortin receptor 4(Homo sapiens (Human))
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250586(CHEMBL4093140)
Affinity DataIC50:  0.400nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250586(CHEMBL4093140)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed