Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1A' and Ligand = 'BDBM50086001'
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50086001(CHEMBL274438 | N-[2-(11-Methoxy-6,7-dihydro-5H-ben...)
Affinity DataKi:  66nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50086001(CHEMBL274438 | N-[2-(11-Methoxy-6,7-dihydro-5H-ben...)
Affinity DataKi:  66nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to human melatonin receptor type 1A (MT1) expressed in NIH3T3 rat fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50086001(CHEMBL274438 | N-[2-(11-Methoxy-6,7-dihydro-5H-ben...)
Affinity DataKi:  66nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50086001(CHEMBL274438 | N-[2-(11-Methoxy-6,7-dihydro-5H-ben...)
Affinity DataKi:  66.1nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed