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Found 4 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1B' and Ligand = 'BDBM50240442'
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50240442(CHEMBL33185 | N-((1-(4-chlorobenzyl)-4-methoxy-1H-...)
Affinity DataKi:  8.70nMAssay Description:Antagonist activity at human MT2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50240442(CHEMBL33185 | N-((1-(4-chlorobenzyl)-4-methoxy-1H-...)
Affinity DataKi:  8.70nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to human melatonin receptor MT2 expressed in NIH3T3 rat fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50240442(CHEMBL33185 | N-((1-(4-chlorobenzyl)-4-methoxy-1H-...)
Affinity DataKi:  8.70nMAssay Description:Binding affinity towards melatonin receptor type 1B stably expressed in NIH3T3 rat fibroblast cells using 2-[125I]iodomelatoninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50240442(CHEMBL33185 | N-((1-(4-chlorobenzyl)-4-methoxy-1H-...)
Affinity DataKi:  9nMAssay Description:Displacement of 2-[125I]Iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed