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Found 2 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 1' and Ligand = 'BDBM50058047'
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058047(CHEMBL3330812 | US9260448, 29)
Affinity DataIC50:  74nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058047(CHEMBL3330812 | US9260448, 29)
Affinity DataIC50:  74nMAssay Description:Cells of Chem3 Cell Line (HTS145C:Millipore) in which mGluR1 was stably expressed were adjusted to a density of 2×106/ml. 50 μl of the cells wer...More data for this Ligand-Target Pair
In DepthDetails US Patent