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Found 1 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 5' and Ligand = 'BDBM109116'
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM109116(US8609852, 23)
Affinity DataKi:  1.60nM ΔG°:  -50.2kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In DepthDetails US Patent