Affinity DataKi: 31nMAssay Description:Displacement of [3H]-aldosterone from rat mineralocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 256nMAssay Description:Antagonist activity at human wild-type mineralocorticoid receptor expressed in CHO-K1 cells assessed as inhibition of aldosterone-induced transcripti...More data for this Ligand-Target Pair
Affinity DataIC50: 276nMAssay Description:Displacement of [3H]-aldosterone from recombinant human mineralocorticoid receptor expressed in baculovirus infected insect cells incubated overnight...More data for this Ligand-Target Pair
Affinity DataIC50: <500nMAssay Description:Binding affinity to rat mineralocorticoid receptorMore data for this Ligand-Target Pair