Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase 1' and Ligand = 'BDBM7491'
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:In vitro inhibitory concentration against human mitogen-activated protein kinase-1 (MEK-1) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of Mitogen-activated protein kinase (MAPK)phosphorylation by activated MEK-1More data for this Ligand-Target Pair