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Found 4 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase 8' and Ligand = 'BDBM50342301'
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342301(2-(2-(benzo[b]thiophen-3-yl)acetamido)thiophene-3-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342301(2-(2-(benzo[b]thiophen-3-yl)acetamido)thiophene-3-...)
Affinity DataIC50:  4.62E+3nMAssay Description:Displacement of biotin-labeled JIP1 peptide from JNK1 by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342301(2-(2-(benzo[b]thiophen-3-yl)acetamido)thiophene-3-...)
Affinity DataKd:  3.10E+3nMAssay Description:Binding affinity to JNK1 in presence of peptide JIP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342301(2-(2-(benzo[b]thiophen-3-yl)acetamido)thiophene-3-...)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to JNK1 in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed