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Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 12' and Ligand = 'BDBM365261'
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM365261(2-Imidazol-1-yl-1-{3-[2- (2-methyl-pyrrolidin-1- y...)
Affinity DataKi:  1.59nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM365261(2-Imidazol-1-yl-1-{3-[2- (2-methyl-pyrrolidin-1- y...)
Affinity DataKi:  7.69nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent