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Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 20' and Ligand = 'BDBM50268010'
TargetMitogen-activated protein kinase kinase kinase 20(Homo sapiens (Human))
University Of Macau

Curated by ChEMBL
LigandPNGBDBM50268010(CHEMBL4098896)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full-length ZAK expressed in baculovirus infected Sf9 insect cells using MBP as substrate after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 20(Homo sapiens (Human))
University Of Macau

Curated by ChEMBL
LigandPNGBDBM50268010(CHEMBL4098896)
Affinity DataKd:  2.70nMAssay Description:Binding affinity to partial length human ZAK expressed in Escherichia coli BL21 by active-site-dependent competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed