Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase kinase 2' and Ligand = 'BDBM43248'
LigandPNGBDBM43248((5Z)-5-[(2E)-2-(3-ethyl-4,5-diphenyl-1,3-thiazol-2...)
Affinity DataEC50:  2.73E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
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LigandPNGBDBM43248((5Z)-5-[(2E)-2-(3-ethyl-4,5-diphenyl-1,3-thiazol-2...)
Affinity DataEC50:  3.22E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay